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Classification

FDA Approved Peptides

FDA Approved

Peptide medicines that have completed FDA review and carry an approved label for one or more specific uses. These are prescription products dispensed through licensed pharmacies under physician supervision.

AI Summary

FDA Approved Peptides on Peptides.cafe are approved by the u.s. fda for one or more specific indications. This hub lists 70 peptides in this classification, each with a mechanism of action, commonly researched wellness goals, a research summary, safety considerations, and primary references. Classification is educational and describes regulatory status only — it is not medical advice and does not indicate suitability for any individual.

All fda approved peptides (70)

Abaloparatide (Tymlos)Clinical

PTHrP analog for postmenopausal osteoporosis.

Anidulafungin (Eraxis)Clinical

Echinocandin lipopeptide for invasive Candida infections.

Bivalirudin (Angiomax)Clinical

Direct thrombin inhibitor peptide for PCI anticoagulation.

Bremelanotide (Vyleesi)Hormonal

Melanocortin receptor agonist for hypoactive sexual desire disorder in premenopausal women.

Calcitonin-Salmon (Miacalcin)Clinical

32-amino-acid peptide for osteoporosis and hypercalcemia.

Caspofungin (Cancidas)Clinical

Echinocandin lipopeptide for invasive Candida and Aspergillus infections.

Cetrorelix (Cetrotide)Clinical

GnRH antagonist used in IVF to prevent premature ovulation.

Colistin (Polymyxin E)Clinical

Last-resort lipopeptide antibiotic for multidrug-resistant Gram-negatives.

Corticorelin (Acthrel)Clinical

Synthetic ovine CRH for differential diagnosis of Cushing's syndrome.

Cosyntropin (Cortrosyn)Clinical

Synthetic ACTH(1-24) for adrenal function testing.

Dalbavancin (Dalvance)Clinical

Long-acting lipoglycopeptide for skin and soft tissue infections.

Daptomycin (Cubicin)Clinical

Cyclic lipopeptide antibiotic for serious Gram-positive infections.

Degarelix (Firmagon)Hormonal

GnRH antagonist providing immediate testosterone suppression in prostate cancer.

Desmopressin (DDAVP)Clinical

Synthetic vasopressin analog for diabetes insipidus and nocturnal enuresis.

Dulaglutide (Trulicity)Fat loss

Once-weekly GLP-1 agonist with cardiovascular benefit.

Ecallantide (Kalbitor)Clinical

Plasma kallikrein inhibitor for hereditary angioedema.

Enfuvirtide (Fuzeon)Clinical

First-in-class HIV fusion inhibitor peptide.

Eptifibatide (Integrilin)Clinical

GP IIb/IIIa inhibitor cyclic peptide for ACS and PCI.

Etelcalcetide (Parsabiv)Clinical

Calcimimetic peptide for secondary hyperparathyroidism on hemodialysis.

Exenatide (Byetta / Bydureon)Fat loss

First-in-class GLP-1 receptor agonist for type 2 diabetes.

Ganirelix (Antagon)Clinical

GnRH antagonist for IVF cycles.

Glatiramer Acetate (Copaxone)Cognitive

Synthetic random peptide copolymer for relapsing multiple sclerosis.

Glucagon (GlucaGen / Baqsimi)Hormonal

29-amino-acid peptide hormone for severe hypoglycemia.

Goserelin (Zoladex)Hormonal

GnRH agonist implant for hormone-sensitive cancers.

Histrelin (Supprelin LA / Vantas)Hormonal

GnRH agonist implant for central precocious puberty and prostate cancer.

Icatibant (Firazyr)Clinical

Bradykinin B2 receptor antagonist for hereditary angioedema attacks.

Insulin Aspart (NovoLog)Hormonal

Rapid-acting mealtime insulin analog.

Insulin Degludec (Tresiba)Hormonal

Ultra-long-acting basal insulin with >42-hour duration.

Insulin Glargine (Lantus)Hormonal

Long-acting basal insulin analog for type 1 and type 2 diabetes.

Insulin Lispro (Humalog)Hormonal

Rapid-acting mealtime insulin analog.

Lanreotide (Somatuline)Clinical

Long-acting somatostatin analog for acromegaly and NETs.

Leuprolide (Lupron)Hormonal

GnRH agonist used for prostate cancer, endometriosis, and precocious puberty.

Linaclotide (Linzess)Clinical

Guanylate cyclase-C agonist peptide for IBS-C and chronic constipation.

LiraglutideFat loss

FDA-approved daily GLP-1 receptor agonist.

Lixisenatide (Adlyxin)Fat loss

Short-acting GLP-1 agonist focused on postprandial glucose.

Lonapegsomatropin (Skytrofa)Performance

Long-acting pegylated growth hormone, once-weekly.

Macimorelin (Macrilen)Clinical

Oral ghrelin agonist for diagnosing adult growth hormone deficiency.

MazdutideFat loss

GLP-1/glucagon dual agonist in Phase 3 development.

Mecasermin (Increlex)Performance

Recombinant human IGF-1 for severe primary IGF-1 deficiency.

Micafungin (Mycamine)Clinical

Echinocandin antifungal for Candida infections and prophylaxis.

Motixafortide (Aphexda)Clinical

CXCR4 antagonist peptide that mobilizes stem cells for autologous transplant in multiple myeloma.

Nafarelin (Synarel)Hormonal

Intranasal GnRH agonist for endometriosis and central precocious puberty.

Nesiritide (Natrecor)Clinical

Recombinant BNP for acute decompensated heart failure.

Octreotide (Sandostatin)Clinical

Synthetic somatostatin analog for acromegaly and neuroendocrine tumors.

Oritavancin (Orbactiv / Kimyrsa)Clinical

Single-dose lipoglycopeptide for acute bacterial skin and skin structure infections.

OxytocinCognitive

Neuropeptide studied for social bonding and stress modulation.

Pasireotide (Signifor)Clinical

Multi-receptor somatostatin analog for Cushing's disease and acromegaly.

Pegvisomant (Somavert)Clinical

Pegylated GH receptor antagonist for acromegaly.

Plecanatide (Trulance)Clinical

Uroguanylin analog for chronic constipation.

Pramlintide (Symlin)Fat loss

Amylin analog adjunct to mealtime insulin.

PT-141 (Bremelanotide)Hormonal

Melanocortin agonist researched for sexual desire and arousal.

Rezafungin (Rezzayo)Clinical

Once-weekly echinocandin for candidemia and invasive candidiasis.

Romiplostim (Nplate)Clinical

Thrombopoietin-receptor peptibody for immune thrombocytopenia.

SemaglutideFat loss

FDA-approved GLP-1 agonist for diabetes and obesity.

Setmelanotide (Imcivree)Clinical

MC4R agonist for rare genetic obesity disorders.

Sincalide (Kinevac)Clinical

Synthetic C-terminal octapeptide of cholecystokinin for gallbladder imaging.

Somapacitan (Sogroya)Performance

Once-weekly growth hormone analog for adults and children with GHD.

Somatrogon (Ngenla)Performance

Long-acting recombinant human growth hormone for pediatric GH deficiency — weekly dosing.

Synthetic Secretin (ChiRhoStim)Clinical

27-amino-acid peptide used to stimulate pancreatic secretions for diagnosis.

Teduglutide (Gattex)Clinical

GLP-2 analog for short bowel syndrome dependent on parenteral support.

Telavancin (Vibativ)Clinical

Lipoglycopeptide for complicated skin infections and HABP/VABP.

Teriparatide (Forteo)Clinical

Recombinant PTH(1-34) for severe osteoporosis.

TesamorelinPerformance

GHRH analog FDA-approved for HIV-associated visceral fat.

TirzepatideFat loss

FDA-approved GLP-1/GIP dual agonist.

Triptorelin (Trelstar)Clinical

GnRH agonist depot for advanced prostate cancer.

VancomycinClinical

Glycopeptide antibiotic for serious Gram-positive infections including MRSA.

Vasopressin (Vasostrict)Clinical

Nonapeptide hormone used for vasodilatory shock.

Vosoritide (Voxzogo)Clinical

C-type natriuretic peptide analog for achondroplasia.

Ziconotide (Prialt)Clinical

Synthetic ω-conopeptide for severe chronic pain via intrathecal infusion.

Zilucoplan (Zilbrysq)Cognitive

Macrocyclic peptide complement C5 inhibitor for generalized myasthenia gravis.

Frequently asked questions

What makes a peptide FDA approved?

An FDA-approved peptide has completed the agency's review process and carries an approved label describing the indication, dosing, and safety information supported by clinical trial data. Approval applies to the specific product and indication reviewed, not to the peptide molecule in every possible use.

How many FDA approved peptides are covered in this library?

Peptides.cafe currently documents 70 peptides with an approved FDA label, each with a mechanism overview, commonly researched wellness goals, safety considerations, and primary references.

Are FDA approved peptides available without a prescription?

No. FDA-approved peptide medicines are prescription products dispensed through licensed pharmacies under the supervision of a licensed healthcare provider.

Is an FDA approved peptide safer than a compounded or research peptide?

FDA-approved products have been evaluated for manufacturing quality, purity, and labelled safety in clinical trials, which compounded and research peptides have not. That does not make any product risk-free — every peptide has a safety profile that should be reviewed with a licensed clinician.

Other classifications

Educational Wellness Information Only

This platform provides peer-reviewed research summaries and educational content about peptides for wellness and optimization purposes. Nothing on this site is intended as medical advice, diagnosis, or treatment. We do not claim any peptide can diagnose, treat, cure, or prevent any disease. Always consult a licensed healthcare provider before beginning any wellness protocol.

Statements on this site have not been evaluated by the FDA. Compounded preparations are subject to applicable state and federal regulations. Availability and eligibility vary.